203297
Bisindolylmaleimide IV
Arcyriarubin A, 2,3-bis(1H-Indol-3-yl)maleimide, Ro 31-6233
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Merck KGaA
Frankfurter Str. 250
64293 Darmstadt
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Fax: +49 6151 72 2000
15 February 2012
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A potent, cell permeable, and selective inhibitor of protein kinase C (IC50 = 87 nM). Inhibits protein kinase A at much higher concentrations (IC50 = 2.7 µM).
| Product information | |||
|---|---|---|---|
| Form | Orange solid | ||
| Primary Target | PKC | ||
| Primary Target IC50 | 87 nM | ||
| Secondary target | PKA (IC50 = 2.7 µM) | ||
| Molar mass | 327.3 | ||
| Cell permeable | Yes | ||
| Purity | ≥95% by HPLC | ||
| Solubility | DMSO or MeOH | ||
| Chemical formula | C20H13N3O2 | ||
| CAS number | 119139-23-0 | ||
| Store and ship information | |||
|---|---|---|---|
| Storage | +2°C to +8°C | ||
| Ship |
Ambient Temperature Only
Standard Handling |
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