100122
A3, Hydrochloride
N-(2-Aminoethyl)-5-chloronaphthalene-1-sulfonamide, HCl
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15 February 2012
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A cell-permeable, reversible, and shorter alkyl chain derivative of W-7 that inhibits casein kinase I (Ki = 80 µM), casein kinase II (Ki = 5.1 µM), myosin light chain kinase (Ki = 7.4 µM), protein kinase A (Ki = 4.3 µM), protein kinase C (Ki = 47 µM), and protein kinase G (Ki = 3.8 µM).
| Product information | |||
|---|---|---|---|
| Form | Off-white solid | ||
| Primary Target | CK1 | ||
| Primary Target Ki | 80 µM | ||
| Secondary target | CK2 (Ki = 5.1 µM), MLCK (Ki = 7.4 µM), PKA (Ki = 4.3 µM), PKC (Ki = 47 µM), PKG (Ki = 3.8 µM) | ||
| Molar mass | 321.2 | ||
| Hygrocopic | Yes | ||
| Purity | ≥98% by TLC | ||
| Solubility | DMSO or 50% Ethanol | ||
| Chemical formula | C12H13ClN2O2S · HCl | ||
| CAS number | 78957-85-4 | ||
| Store and ship information | |||
|---|---|---|---|
| Storage | -20°C | ||
| Ship |
Ambient Temperature Only
Standard Handling |
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