Cell permable and less potent than H-7 in inhibiting rat brain protein kinase C isoforms (IC50 = 50 µM). Also inhibits cyclic-nucleotide-dependent protein kinases.
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Product information
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Form
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Faint yellow lyophilized solid
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Primary Target
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PKC isoforms
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Primary Target IC50
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50 µM
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Molar mass
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364.3
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Protect from Light
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Yes
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Packaged under inert gas
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Yes
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Cell permeable
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Yes
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Purity
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≥98% by TLC
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Solubility
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H2O
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Chemical formula
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C14H17N3O2S · 2HCl
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CAS number
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140663-38-3
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Store and ship information
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Storage
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+2°C to +8°C
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Ship
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Ambient Temperature Only
Standard Handling
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