A potent, cell permeable, and selective inhibitor of protein kinase C (IC50 = 87 nM). Inhibits protein kinase A at much higher concentrations (IC50 = 2.7 µM).
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Product information
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Form
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Orange solid
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Primary Target
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PKC
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Primary Target IC50
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87 nM
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Secondary target
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PKA (IC50 = 2.7 µM)
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Molar mass
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327.3
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Cell permeable
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Yes
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Purity
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≥95% by HPLC
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Solubility
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DMSO or MeOH
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Chemical formula
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C20H13N3O2
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CAS number
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119139-23-0
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Store and ship information
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Storage
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+2°C to +8°C
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Ship
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Ambient Temperature Only
Standard Handling
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